Ara mostrant els elements 1-7 de 7
Granados Ramírez, Carmen Giovana (Data de defensa: 2008-01-16)
1) "Diseño, síntesis y caracterización de inhibidores de la fusión de VIH-1 análogos del péptido C34 de gp41 con D aminoácido"<br/><br/>En el proceso de fusión del virus del VIH-1 a la célula diana ...
Martinell Pedemonte, Marc (Data de defensa: 2004-03-29)
En la majoria de processos cel·lulars, hi ha multitud de proteïnes que interaccionen entre sí, essent aquests contactes proteïna-proteïna, fonamentals per al correcte funcionament de cadascun d'aquests ...
Garcia Pindado, Júlia (Data de defensa: 2017-05-12)
The present thesis is based on the development and optimization of a solid-phase strategy to prepare biaryl bicyclic pentapeptides. Suzuki-Miyaura cross-coupling reactions were used to obtain the biaryl ...
Guardiola Bagán, Salvador (Data de defensa: 2017-09-15)
Protein-protein interactions (PPIs) and protein surfaces are considered challenging targets for drug discovery. In this field, conventional medicinal chemistry (i.e. small molecules) has largely failed ...
Pastor Porras, José Javier (Data de defensa: 2004-05-03)
En la presente tesis doctoral se ha desarrollado una nueva estrategia de química combinatoria para la modificación de la hélice alfa C-terminal del dominio B de la proteína A de <i>Staphylococcus ...
Díaz Perlas, Cristina (Data de defensa: 2018-03-07)
Peptides play a critical role in human physiology and harbour a huge potential as therapeutic agents. In this thesis, new peptides have been discovered as ligands for the epidermal growth factor (EGF) ...
Ciudad Fernández, Sonia (Data de defensa: 2016-11-08)
The present thesis is based on the work developed about the use of peptides and small proteins in protein surface molecular recognition. Peptides present several advantages when compared with small ...